2. Vitamin D Related/Nuclear Receptor Metabolic Enzyme/Protease
  3. Progesterone Receptor Androgen Receptor Phosphatase
  4. Trimegestone

Trimegestone  (Synonyms: RU 27987)

目录号: HY-106827
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摩尔计算器

Trimegestone (RU 27987) 是一种具有口服活性的去甲孕酮孕激素。Trimegestone 与孕酮受体 (PR) 结合，IC50 值为 3.3 nM (大鼠 PR)。Trimegestone 还增加碱性磷酸酶活性 (EC50=0.1 nM)，但不增加荧光素酶活性。Trimegestone 还表现出弱的抗雄激素活性 (弱雄激素受体亲和力)。Trimegestone 可用于避孕药或更年期综合征的研究。

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Trimegestone Chemical Structure

Trimegestone Chemical Structure

CAS No. : 74513-62-5

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Trimegestone 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Trimegestone (RU 27987) is an orally active 19-norpregnane progestin. Trimegestone binds to progesterone receptor (PR) with an IC50 value of 3.3 nM (rat PR). Trimegestone increases alkaline phosphatase activity (EC50=0.1 nM) but not luciferase activity. Trimegestone also shows a weak antiandrogenic activity (weak androgen receptor affinity). Trimegestone can be used in studies of contraception or menopausal syndromes[1][2].

Clinical Trial
分子量

342.47

Formula

C22H30O3
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Trimegestone 相关分类

  • 摩尔计算器

  • 稀释计算器

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× = ×
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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Trimegestone74513-62-5RU 27987RU27987RU-27987Progesterone ReceptorAndrogen ReceptorPhosphataseNR3C3Inhibitorinhibitorinhibit

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