2. GPCR/G Protein Neuronal Signaling
  3. Dopamine Receptor 5-HT Receptor
  4. cis-(Z)-Flupentixol dihydrochloride

cis-(Z)-Flupentixol dihydrochloride  (Synonyms: 盐酸氟哌噻吨; cis-(Z)-Flupenthixol dihydrochloride)

目录号: HY-15856
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cis-(Z)-Flupentixol dihydrochloride 是有效、选择性的多巴胺DA D1/D2 受体的拮抗剂，其对D2 受体和 5-HT2A 的 Ki 值分别为 0.38 nM 和 7 nM。

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cis-(Z)-Flupentixol dihydrochloride

cis-(Z)-Flupentixol dihydrochloride Chemical Structure

CAS No. : 51529-01-2

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Other Forms of cis-(Z)-Flupentixol dihydrochloride:

cis-(Z)-Flupentixol dihydrochloride 相关抗体

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生物活性

cis-(Z)-Flupentixol dihydrochloride is a potent and selective DA D1/D2 receptor antagonist, with Ki values of 0.38 nM and 7 nM for D2 receptor and 5-HT2A, respectively[1][2].

IC50 & Target[2]

5-HT2A Receptor

 

D2 Receptor

0.38 nM (Ki)

5-HT2A Receptor

7 nM (Ki)

体内研究
(In Vivo)

cis-(Z)-Flupentixol (0.25, or 0.5 mg/kg, i.p.) pretreatment dose-dependently reduces cocaine-induced activity[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Rats[1].
Dosage: 0.125, 0.25, or 0.5 mg/kg.
Administration: IP.
Result: Reduced cocaine-induced activity.
分子量

507.44

Formula

C23H27Cl2F3N2OS
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

cis-(Z)-Flupentixol dihydrochloride 相关分类

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

cis-(Z)-Flupentixol51529-01-2cis-(Z)-FlupenthixolDopamine Receptor5-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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