Dopamine Receptor Inhibitors

Dopamine Receptor

D₁ Receptor

D₂ Receptor

D₃ Receptor

D₄ Receptor

D₅ Receptor

Dopamine Receptor Ligands, Inhibitors, Agonists, Antagonists & Modulators

Product Name	Dopamine Receptor	D₁ Receptor	D₂ Receptor	D₃ Receptor	D₄ Receptor	D₅ Receptor	Purity
SCH-23390 hydrochloride		D₁ Receptor, Ki: 0.2 nM				D₅ Receptor, Ki: 0.3 nM	99.83%
Haloperidol			D₂ Receptor				99.73%
Clozapine			D₂ Receptor, Ki: 75 nM (Antagonist)				99.84%
Olanzapine	Dopamine Receptor						99.96%
Risperidone			D₂ Receptor, Ki: 5.9 nM				99.87%
Bromocriptine mesylate			D₂ Receptor				99.98%
SKF 38393 hydrochloride		D₁ Receptor					99.49%
WAY-100635					D₄ Receptor		99.51%
Aripiprazole			D₂ Receptor	D₃ Receptor	D₄ Receptor		99.95%
Sulpiride			D₂ Receptor	D₃ Receptor			99.28%
Brexpiprazole			D_2L Receptor, Ki: 0.3 nM				99.80%
Cabergoline			D₂ Receptor	D₃ Receptor			99.86%
Raclopride		D₁ Receptor, Ki: 18000 nM	D₂ Receptor, Ki: 1.8 nM	D₃ Receptor, Ki: 3.5 nM	D₄ Receptor, Ki: 2400 nM		99.86%
Penfluridol			D₂ Receptor				99.93%
SKF 81297		D₁ Receptor					99.86%
Cariprazine			D₂ Receptor, Ki: 0.49 nM	D₃ Receptor, Ki: 0.085 nM			99.67%
Ritanserin			D₂ Receptor, IC₅₀: 70 nM				99.68%
Domperidone			D₂ Receptor				99.87%
Perphenazine			D₂ Receptor, Ki: 0.56 nM	D₃ Receptor, Ki: 0.43 nM	D₄ Receptor, Ki: 28.5 nM		99.80%
Buspirone			Dopamine D2 receptor				99.86%
Rotigotine		D₁ Receptor, Ki: 83 nM	D₂ Receptor, Ki: 4-15 nM	D₃ Receptor, Ki: 0.71 nM	D₄ Receptor, Ki: 4-15 nM	D₅ Receptor, Ki: 4-15 nM	99.99%
SKF 81297 hydrobromide		D₁ Receptor					99.62%
Ropinirole hydrochloride			D₂ Receptor, Ki: 29 nM hD₂ Receptor, pEC₅₀: 7.4	hD₃ Receptor, pEC₅₀: 8.4	hD_4.4 Receptor, pEC₅₀: 6.8		99.89%
N-Methyldopamine hydrochloride		D₁ Receptor					99.12%
Cariprazine hydrochloride			D₂ Receptor, Ki: 0.49 nM	D₃ Receptor, Ki: 0.085 nM			99.88%
Ziprasidone			Rat D₂ Receptor, Ki: 4.8 nM				99.35%
Nuciferine			D₂ Receptor, EC₅₀: 64 nM		D₄ Receptor, EC₅₀: 2 μM	D₅ Receptor, EC₅₀: 2.6 μM	99.90%
Paliperidone			D₂ Receptor				99.43%
WAY-100635 maleate					D₄ Receptor		99.57%
Benztropine mesylate			Human D₂ Receptor				99.85%
Amisulpride			Human D₂ Receptor, Ki: 2.8 nM	D₃ Receptor, Ki: 3.2 nM			99.81%
Rotigotine Hydrochloride		D₁ Receptor, Ki: 83 nM	D₂ Receptor, Ki: 4-15 nM	D₃ Receptor, Ki: 0.71 nM	D₄ Receptor, Ki: 4-15 nM	D₅ Receptor, Ki: 4-15 nM	99.45%
Sumanirole maleate			D₂ Receptor				99.78%
SKF-82958 hydrobromide		D₁ Receptor					99.82%
Loxapine succinate		Human D₁ Receptor	Human D₂ Receptor		Human D₄ Receptor		98.84%
L-741626					D₄ Receptor		99.0%
Lurasidone			D₂ Receptor, IC₅₀: 1.68 nM				99.36%
Dihydrexidine hydrochloride		D₁ Receptor, IC₅₀: 10 nM					98.89%
Flunarizine dihydrochloride			D₂ Receptor				99.36%
Pramipexole			D₂ Receptor, Ki: 3.9 nM	D₃ Receptor, Ki: 0.5 nM	D₄ Receptor, Ki: 1.3 nM		99.88%
Rotundine		D₁ Receptor, IC₅₀: 166 nM	D₂ Receptor, IC₅₀: 1400 nM	D₃ Receptor, IC₅₀: 3300 nM			99.96%
Blonanserin		D₁ Receptor, Ki: 1070 nM	D₂ Receptor, Ki: 0.142 nM	D₃ Receptor, Ki: 0.494 nM	D₄ Receptor, Ki: 150 nM		99.62%
Pramipexole dihydrochloride			D₂ Receptor	D₃ Receptor	D₄ Receptor		99.73%
Loxapine		Human D₁ Receptor	Human D₂ Receptor		Human D₄ Receptor		99.93%
Metoclopramide			D₂ Receptor, IC₅₀: 483 nM				99.98%
Flupentixol dihydrochloride		D₁ Receptor	D₂ Receptor				99.73%
Flunarizine			D₂ Receptor				99.93%
Eticlopride hydrochloride			D₂ Receptor, Ki: 0.09 nM				99.45%
A68930 hydrochloride		D₁ Receptor					98.71%
Ecopipam hydrochloride		D₁ Receptor, Ki: 1.2 nM	D₂ Receptor, Ki: 980 nM		D₄ Receptor, Ki: 5520 nM	D₅ Receptor, Ki: 2.0 nM	99.46%
SKF-83566		D₁ Receptor				D₅ Receptor	99.86%
Pridopidine			D₂ Receptor				99.85%
Piribedil			D₂ Receptor	D₃ Receptor			99.92%
LY3154207		D₁ Receptor					98.06%
Lumateperone		D₁ Receptor	D₂ Receptor				99.83%
Lisuride			D₂ Receptor				99.85%
L-745870			D₂ Receptor, Ki: 960 nM	D₃ Receptor, Ki: 2300 nM	Human D₄ Receptor, Ki: 4.3 nM		99.92%
Talipexole dihydrochloride			D₂ Receptor				99.80%
Bromperidol			D₂ Receptor				99.83%
Pergolide mesylate		D₁ Receptor	D₂ Receptor				99.98%
Thiethylperazine			D₂ Receptor				99.91%
Iloperidone		Rat D₁ Receptor, Ki: 546 nM Human D₁ Receptor, Ki: 216 nM	Rat D₂ Receptor, Ki: 54 nM	Human D₃ Receptor, Ki: 7.1 nM	Human D₄ Receptor, Ki: 25 nM	Human D₅ Receptor, Ki: 319 nM	99.93%
Chlorprothixene		Human D₁ Receptor, Ki: 18 nM	Human D₂ Receptor, Ki: 2.96 nM	Human D₃ Receptor, Ki: 4.56 nM		Human D₅ Receptor, Ki: 9 nM	99.87%
SB-277011 hydrochloride				D₃ Receptor, Ki: 10.7-11.2 nM			99.59%
UNC9994 hydrochloride		D₁ Receptor, Ki: 4000 nM	D₂ Receptor, Ki: 79 nM	D₃ Receptor, Ki: 17 nM	D₄ Receptor, Ki: 138 nM		99.50%
UNC9995			D₂ Receptor				99.93%
Paliperidone palmitate			D₂ Receptor				99.93%
UCSF924					D₄ Receptor		99.53%
Zuclopenthixol			D₂ Receptor				98.08%
Chlorprothixene hydrochloride		Human D₁ Receptor, Ki: 18 nM	Human D₂ Receptor, Ki: 2.96 nM	Human D₃ Receptor, Ki: 4.56 nM		Human D₅ Receptor, Ki: 9 nM	99.91%
Asenapine		D₁ Receptor, pKi: 8.9	D₂ Receptor, pKi: 8.9	D₃ Receptor, pKi: 9.4	D₄ Receptor, pKi: 9.0		99.62%
Lurasidone Hydrochloride			D₂ Receptor, IC₅₀: 1.68 nM				99.86%
Promazine hydrochloride			D₂ Receptor				99.87%
Itopride hydrochloride			D₂ Receptor				99.84%
Lumateperone tosylate		D₁ Receptor	D₂ Receptor				99.78%
PD-168077 maleate					D₄ Receptor		99.60%
Ziprasidone hydrochloride monohydrate			Rat D₂ Receptor, Ki: 4.8 nM				98.11%
Ansofaxine hydrochloride	Dopamine Receptor, IC₅₀: 491 nM						99.72%
Pericyazine			D₂ Receptor				99.86%
SKF 83959		D₁ Receptor, Ki: 1.18 nM	D₂ Receptor, Ki: 920 nM	D₃ Receptor, Ki: 399 nM		D₅ Receptor, Ki: 7.56 nM
Metopimazine			D₂ Receptor				99.75%
GSK598809				D₃ Receptor			99.74%
Pramipexole dihydrochloride hydrate			D₂ Receptor, Ki: 3.9 nM	D₃ Receptor, Ki: 0.5 nM	D₄ Receptor, Ki: 1.3 nM		98.0%
Dehydroaripiprazole			D₂ Receptor	D₃ Receptor			99.95%
Metoclopramide hydrochloride hydrate			D₂ Receptor, IC₅₀: 483 nM				99.96%
Fluphenazine decanoate			D₂ Receptor				98.75%
(+)-PD 128907 hydrochloride			D₂ Receptor	D₃ Receptor			98.92%
Tiapride hydrochloride			D₂ Receptor, IC₅₀: 110-320 nM	D₃ Receptor, IC₅₀: 180 nM			99.95%
Oxypertine			D₂ Receptor, Ki: 30 nM				99.84%
L-DOPA-2,5,6-d₃				D₃ Receptor			98.80%
SKF 83822		Rat D₁ Receptor					98.01%
GR 103691				D₃ Receptor			99.91%
Brilaroxazine			D₂ Receptor	D₃ Receptor	D₄ Receptor		98.82%
Xaliproden hydrochloride			D₂ Receptor, IC₅₀: 0.1-1 μM				98.57%
Spiperone hydrochloride		D₁ Receptor, Ki: ~350 nM	D₂ Receptor, Ki: 0.06 nM	D₃ Receptor, Ki: 0.6 nM	D₄ Receptor, Ki: 0.08 nM	D₅ Receptor, Ki: ~3500 nM	99.10%
Halopemide		D₁ Receptor	D₂ Receptor				99.65%
Nemonapride			D₂ Receptor, Ki: 0.06 nM				99.90%
(Rac)-Tavapadon		D₁ Receptor					99.87%
Sarizotan			rD₂ Receptor, IC₅₀: 15.1 nM (rat) hD₂ Receptor, IC₅₀: 17 nM	D₃ Receptor, IC₅₀: 6.8 nM (human)	hD_4.2 Receptor, IC₅₀: 2.4 nM		98.23%
Desmethyl cariprazine			D₂ Receptor, Ki: 0.49 nM	D₃ Receptor, Ki: 0.085 nM			98.08%
Propionylpromazine hydrochloride			D₂ Receptor				99.71%
NGB 2904				D₃ Receptor, Ki: 1.4 nM			98.28%
Ocaperidone			D₂ Receptor, Ki: 0.75 nM				99.93%
Pipamperone			D₂ Receptor, pKi: 6.7		D₄ Receptor, pKi: 8.0		99.89%
L-745870 hydrochloride			D₂ Receptor, Ki: 960 nM	D₃ Receptor, Ki: 2300 mM	Human D₄ Receptor, Ki: 4.3 nM		99.91%
Amisulpride hydrochloride				D₃ Receptor			99.79%
CY 208-243		D₁ Receptor					99.99%
ML417				D₃ Receptor, EC₅₀: 38 nM			99.50%
Dopamine D4 receptor antagonist-1					hD_4.2 Receptor, Ki: 9.0 nM		98.59%
Melperone			Human D₂ Receptor, Kd: 180 nM				99.84%
Perospirone hydrochloride		D₁ Receptor, Ki: 41 nM	D₂ Receptor, Ki: 1.4 nM				99.94%
UNC9994			D₂ Receptor, Ki: 79 nM	D₃ Receptor, Ki: 17 nM	D₄ Receptor, Ki: 138 nM		98.06%
Didesmethyl cariprazine			D_2L Receptor, Ki: 1.41 nM	Human D₃ Receptor, Ki: 0.056 nM			99.63%
Ecopipam		D₁ Receptor, Ki: 1.2 nM	D₂ Receptor, Ki: 980 nM		D₄ Receptor, Ki: 5520 nM	D₅ Receptor, Ki: 2.0 nM	99.77%
Sonepiprazole			rD₂ Receptor, Ki: 5147 nM		rD₄ Receptor, Ki: 3.6 nM		98.43%
Olanzapine-d₃				D₃ Receptor			99.09%
PF-06256142		Human D₁ Receptor, EC₅₀: 33 nM					99.90%
LE 300		Human D₁ Receptor, Ki: 1.9 nM				Human D₅ Receptor, Ki: 7.5 nM	98.5%
D5R agonist 1						D₅ Receptor, EC₅₀: 269.7 nM	99.83%
Neuromedin N			D₂ Receptor				99.84%
Roxindole hydrochloride			D₂ Receptor				99.48%
Naxagolide			D₂ Receptor				99.81%
Adoprazine			D₂ Receptor, pA2: 9.3 D₂ Receptor, pKi: 8.4	D₃ Receptor, pA2: 8.9 D₃ Receptor, pKi: 8.4	D₄ Receptor, pKi: 8.0		98.60%
L-Stepholidine		D₁ Receptor	D₂ Receptor				99.41%
Quinelorane dihydrochloride			D₂ Receptor	D₃ Receptor			99.0%
NGD94-1					hD_4.2 Receptor, Ki: 3.6 nM		99.73%
(Rac)-PF-06256142		Human D₁ Receptor, EC₅₀: 107 nM					99.59%
Brexpiprazole S-oxide-d₈			D₂ Receptor, Ki: 0.3 nM				98.72%
A-381393				D₃ Receptor	D₄ Receptor		99.92%
Ziprasidone hydrochloride			Rat D₂ Receptor, Ki: 4.8 nM				99.74%
PAOPA			D₂ Receptor				98.09%
Thioridazine-d₃ hydrochloride				D₃ Receptor			98.25%
Ro 10-5824 dihydrochloride					D₄ Receptor		99.86%
Spiramide		D₁ Receptor, Ki: 2530 nM	D₂ Receptor, Ki: 3 nM				99.23%
Acetophenazine dimaleate			D₂ Receptor				99.90%
Esamisulpride			D₂ Receptor	D₃ Receptor			99.04%
A-77636 hydrochloride			D₂ Receptor				≥98.0%
ABT-724 trihydrochloride					D₄ Receptor		99.05%
Bromopride			D₂ Receptor				99.87%
SKF 83959 hydrobromide		D₁ Receptor, Ki: 1.18 nM	D₂ Receptor, Ki: 920 nM	D₃ Receptor, Ki: 399 nM		D₅ Receptor, Ki: 7.56 nM	99.86%
PG01037 dihydrochloride				D₃ Receptor, Ki: 0.7 nM			99.35%
Pardoprunox hydrochloride			D₂ Receptor, pEC₅₀: 8	D₃ Receptor, pEC₅₀: 9.2			99.46%
Zuclopenthixol-d₄ succinate			D₂ Receptor				99.0%
Ecopipam hydrobromide		D₁ Receptor, Ki: 1.2 nM	D₂ Receptor, Ki: 980 nM		D₄ Receptor, Ki: 5520 nM	D₅ Receptor, Ki: 2.0 nM	99.0%
Aramisulpride			D₂ Receptor, Ki: 140 nM	D₃ Receptor, Ki: 13.9 nM			99.49%
(Rac)-Levomepromazine-d₃ hydrochloride				D₃ Receptor
Mesdopetam				D₃ Receptor
Metoclopramide hydrochloride			D₂ Receptor, IC₅₀: 483 nM				99.96%
Amisulpride-d₅				D₃ Receptor			98.83%
Risperidone-d₄			D₂ Receptor				99.40%
U-99194 maleate				D₃ Receptor, Ki: 160 nM			99.23%
Clomipramine-d₃ hydrochloride				D₃ Receptor			99.98%
Cariprazine-d₈				D₃ Receptor			99.51%
Zuclopenthixol dihydrochloride			D₂ Receptor				99.98%
Haloperidol-d₄			D₂ Receptor
Carmoxirole hydrochloride			D₂ Receptor				99.82%
D3/5-HT receptor modulator-1		D₁ Receptor, Ki: 3290 nM	D₂ Receptor, Ki: 263 nM	D₃ Receptor, Ki: 4.5 nM			99.75%
Benztropine			D₂ Receptor
S-14506 hydrochloride			D₂ Receptor				99.92%
Fananserin					D₄ Receptor, Ki: 2.93 nM		99.97%
SKF-83566 hydrobromide		D₁ Receptor				D₅ Receptor
Thiethylperazine dimaleate			D₂ Receptor				99.99%
CP 226269					D₄ Receptor		99.65%
(-)-GSK598809 hydrochloride				D₃ Receptor			99.64%
cis-(Z)-Flupentixol dihydrochloride			D₂ Receptor, Ki: 0.38 nM
SKF-75670 hydrobromide		D₁ Receptor					99.83%
Brexpiprazole S-oxide			D₂ Receptor, Ki: 0.3 nM
Aripiprazole monohydrate			D₂ Receptor	D₃ Receptor	D₄ Receptor		99.83%
DETQ		Human D₁ Receptor, EC₅₀: 5.8 nM
Asimilobine	Dopamine Receptor						99.9%
Cyclo(glycyl-L-leucyl)	Dopamine Receptor						99.79%
SB-277011 dihydrochloride				D₃ Receptor
FAUC 213			hD₂ Receptor, Ki: 3.4 μM	hD₃ Receptor, Ki: 5.3 μM	hD_4.4 Receptor, Ki: 2.2 nM		99.86%
Moperone			D₂ Receptor, IC₅₀: 1 nM	D₃ Receptor, IC₅₀: 1 nM
ST-836 hydrochloride			D₂ Receptor, Ki: 132 nM	D₃ Receptor, Ki: 4.5 nM
Risperidone hydrochloride			D₂ Receptor, Ki: 5.9 nM
(Rac)-Rotigotine hydrochloride		D₁ Receptor, Ki: 83 nM	D₂ Receptor, Ki: 13.5 nM	D₃ Receptor, Ki: 0.71 nM	D₄ Receptor, Ki: 3.9-15 nM	D₅ Receptor, Ki: 5.4 nM	98.11%
Aplindore			D₂ Receptor, pKi: 9.1				98.44%
5-HT6/7 antagonist 1			D₂ Receptor
Risperidone-d₆			D₂ Receptor, Ki: 5.9 nM
Ziprasidone mesylate trihydrate			Rat D₂ Receptor, Ki: 4.8 nM
Clocapramine			D₂ Receptor
Propionylpromazine-d₆ hydrochloride			D₂ Receptor				99.78%
Blonanserin dihydrochloride		D₁ Receptor, Ki: 1070 nM	D₂ Receptor, Ki: 0.142 nM	D₃ Receptor, Ki: 0.494 nM	D₄ Receptor, Ki: 150 nM
Levosulpiride-d₃				D₃ Receptor			99.79%
Nomifensine-d₃ maleate				D₃ Receptor
Amisulpride-d₅ N-Oxide				D₃ Receptor
Iloperidone-d₃				D₃ Receptor
Cabergoline-d₅			D₂ Receptor	D₃ Receptor
Paliperidone-d₄			D₂ Receptor
Pergolide-d₇ mesylate			D₂ Receptor
Dopamine D3 receptor antagonist-2				D₃ Receptor, Ki: 2.16 nM
D4R antagonist-1					D₄ Receptor, IC₅₀: 6.87 μM
Nooglutil			D₂ Receptor
(-)-IHCH7041			D₂ Receptor, Ki: 22.44 nM
Mesulergine hydrochloride	Dopamine Receptor
Bromocriptine-¹³C,d₃			D₂ Receptor	D₃ Receptor
Razpipadon		D₁ Receptor
Haloperidol-¹³C₆			D₂ Receptor
PF-04363467				D₃ Receptor
D4R antagonist-2					D₄ Receptor
Blonanserin-d₈			D₂ Receptor
Flupenthixol decanoate			D₂ Receptor
Dopamine D4 receptor ligand 2			D₂ Receptor, IC₅₀: >1000 nM		D₄ Receptor, IC₅₀: 0.057 nM
Metopimazine acid-d₆ hydrochloride			D₂ Receptor
N-Methylspiroperidol			D₂ Receptor
Aramisulpride hydrochloride			D₂ Receptor, Ki: 140 nM	D₃ Receptor, Ki: 13.9 nM
Agroclavine		D₁ Receptor
CNV-dopamine			D₂ Receptor
Dopamine D3 receptor antagonist-3				Dopamine D3 receptor, Kd: 0.49 μM
PD 119819	Dopamine Receptor
Carmoxirole			D₂ Receptor
Roxindole			D₂ Receptor
7-Hydroxy-DPAT				D₃ Receptor
Dopamine D2 receptor agonist-3			D₂ Receptor, EC₅₀: 5 nM	D₃ Receptor, EC₅₀: >3.2 μM			98.30%
PD 118717			D₂ Receptor
SV 156			Human D₂ Receptor, Ki: 2.5 ± 0.4 nM	Human D₃ Receptor, Ki: 96.9 ± 4.3 nM	Human D₄ Receptor, Ki: 700 ± 56 nM
A-77636		Dopamine D1 receptor, EC₅₀: 1.1 nM Dopamine D1 receptor, Ki: 39.8 nM
FAUC 346				D₃ Receptor, EC₅₀: 1.5 nM			99.90%
Tau-aggregation-IN-1			D₂ Receptor	D₃ Receptor
Trepipam		D₁ Receptor
BMY 28674			D₂ Receptor, IC₅₀: 3.1 μM	D₃ Receptor, IC₅₀: 4.9 μM	D₄ Receptor, IC₅₀: 0.85 μM
UNC10062		D₁ Receptor
D1/D5 Receptor agonist-1		D₁ Receptor				D₅ Receptor
SK609 hydrochloride				Dopamine D3 receptor, EC₅₀: 1109 nM			99.83%
Fluphenazine decanoate dihydrochloride			D₂ Receptor
Clomipramine-d₃				D₃ Receptor
Ropinirole			D₂ Receptor, Ki: 29 nM hD₂ Receptor, pEC₅₀: 7.4	hD₃ Receptor, pEC₅₀: 8.4	hD_4.4 Receptor, pEC₅₀: 6.8
Dopamine D3 receptor antagonist-1				D₃ Receptor
Dopamine D3 receptor ligand-1			D₂ Receptor, Ki: 715 nM	D₃ Receptor, Ki: 8 nM
OS-3-106				D₃ Receptor, Ki: 0.2 nM
D3R ligand 1				D₃ Receptor, Ki: 66 nM
Iloperidone carboxylic acid		Human D₁ Receptor, pKi: 5.94		Rat D₃ Receptor, pKi: 6.11
Dopamine D2 receptor antagonist-3			D₂ Receptor, pIC₅₀: 5.52
NGB 2904 hydrochloride				D₃ Receptor, Ki: 1.4
Brexpiprazole hydrochloride			D_2L Receptor, Ki: 0.3 nM
MOR agonist-2				D₃ Receptor
Sibenadet			D₂ Receptor
SUN-1334H free base				Dopamine D3 receptor, IC₅₀: 3.43 μM
Acetophenazine			D₂ Receptor				98.05%
BRL 34778			D₂ Receptor, Ki: 2.14 nM
S18327			D₂ Receptor
Perphenazine dihydrochloride			D₂ Receptor, Ki: 0.56 nM	D₃ Receptor, Ki: 0.43 nM	D₄ Receptor, Ki: 28.5 nM
AVE-5997				D₃ Receptor
SKF 38393		D₁ Receptor
Promazine			D₂ Receptor
SSR-181507 hydrochloride			D₂ Receptor
PD 172760					D₄ Receptor
Asenapine citrate		D₁ Receptor, pKi: 8.9	D₂ Receptor, pKi: 8.9	D₃ Receptor, pKi: 9.4	D₄ Receptor, pKi: 9.0
PD 158771			hD₂ Receptor, Ki: 42 nM	Human D₃ Receptor, Ki: 13.7 nM
Cabergoline-d₆			D₂ Receptor	D₃ Receptor
BGC20-761			Human D₂ Receptor, Ki: 140 nM
ARN25657				D₃ Receptor, EC₅₀: 15.2 nM D₃ Receptor, Ki: 1.5 nM
Alizapride-¹³C,d₃ hydrochloride				D₃ Receptor
SKF 38393 hydrobromide		D₁ Receptor, IC₅₀: 110 nM
YM-50001					D₄ Receptor, Ki: 5.62 nM
AL-LAD		D₁ Receptor	D₂ Receptor
D4R antagonis-2					D₄ Receptor, IC₅₀: 6.87 μM
D-520			D₂ Receptor, EC₅₀: 4.73 nM D_2L Receptor, Ki: 41.8 nM	D₃ Receptor, EC₅₀: 2.18 nM D₃ Receptor, Ki: 0.35 nM
A68930		D₁ Receptor
5-HT1AR/5-HT6R ligand-1			D₂ Receptor, Ki: 1903 nM
Dopamine D3 receptor ligand-3			D₂ Receptor, Ki: 353 nM	D₃ Receptor, Ki: 3.6 nM
SCH-23390 maleate		D₁ Receptor, Ki: 0.2 nM				D₅ Receptor, Ki: 0.3 nM
Itopride-d₆ hydrochloride			D₂ Receptor
Piribedil dihydrochloride			D₂ Receptor	D₃ Receptor
Cinitapride monotartrate			D₂ Receptor
Benztropine-¹³C,d₃ mesylate			D₂ Receptor	D₃ Receptor
PD 168568 dihydrochloride			D₂ Receptor, Ki: 1842 nM	D₃ Receptor, Ki: 2682 nM	D₄ Receptor, Ki: 8.8 nM
Ziprasidone mesylate			Rat D₂ Receptor, Ki: 4.8 nM
MLS6357				Dopamine D3 receptor, IC₅₀: 13 μM
Melperone hydrochloride			Human D₂ Receptor, Kd: 180 nM
Dopamine D3 receptor ligand-4			D₂ Receptor, Ki: 7.43 nM	D₃ Receptor, Ki: 0.5 nM
L-750667 triHydrochloride					D₄ Receptor, Ki: 0.51 nM D₄ Receptor, Kd: 0.16 nM		99.39%
Lirexapride			Dopamine D2 receptor
L-745870 trihydrochloride			D₂ Receptor, Ki: 960 nM	D₃ Receptor, Ki: 2300 nM	Human D₄ Receptor, Ki: 4.3 nM
5-HT2A receptor agonist-13			D₂ Receptor, Ki: 1298 nM
(Rac)-Rotigotine-d₇ hydrochloride		D₁ Receptor		D₃ Receptor	D₄ Receptor
Tropapride			D₂ Receptor
SEP-4199			D₂ Receptor
Piquindone			D₂ Receptor
5-HT7R antagonist 3			D₂ Receptor, Ki: 511 nM
Asenapine-¹³C,d₃ hydrochloride				D₃ Receptor	D₄ Receptor
(S)-Remoxipride		D₁ Receptor, IC₅₀: ＞100 μM	D₂ Receptor, IC₅₀: 1.57 μM
PD 168568			D₂ Receptor, Ki: 1842 nM	D₃ Receptor, Ki: 2682 nM	D₄ Receptor, Ki: 8.8 nM
Itopride			D₂ Receptor
PF-4363467			D₂ Receptor, Ki: 692 nM	D₃ Receptor, Ki: 3.1 nM
NGD 94-1 dimaleate					hD_4.2 Receptor, Ki: 3.6 nM
Pramipexole-d₇ dihydrochloride			D₂ Receptor	D₃ Receptor	D₄ Receptor
U-99194				D₃ Receptor
FGH31					Dopamine D4 receptor, Ki: 1.6 nM
Ordopidine			D₂ Receptor
5-HT1AR agonist 2			D₂ Receptor, Ki: 23 nM
Piribedil hydrochloride			D₂ Receptor	D₃ Receptor
NEO 376	Dopamine Receptor						99.23%
Loxapine hydrochloride		Human D₁ Receptor	Human D₂ Receptor		Human D₄ Receptor
UNC9815		D₁ Receptor
D1R antagonist 2		D₁ Receptor, IC₅₀: 35.6 ( cAM nM D₁ Receptor, IC₅₀: 70 (β-arre nM
PNU-177864 hydrochloride				D₃ Receptor
UCSF34			D_2L Receptor, pKi: 7.49
Bromperidol hydrochloride			D₂ Receptor				99.96%
Bifeprunox			D₂ Receptor, pKi: 8.83 (striatum)
PD-143188			D₂ Receptor, Ki: 25.5 nM	D₃ Receptor, Ki: 16.6 nM	hD_4.2 Receptor, Ki: 90.9 nM
Antipsychotic agent-2			D₂ Receptor, Kb: 45.7 nM
BP 897			D₂ Receptor	D₃ Receptor
RU-24213 hydrochloride			Dopamine D2 receptor
A-69024		D₁ Receptor, Ki: 12.6 nM	D₂ Receptor, Ki: 1290 nM
Dopamine D3 receptor ligand-2			D₂ Receptor, Ki: 1228 nM	D₃ Receptor, Ki: 11.4 nM
SKF83822 hydrobromide		D₁ Receptor
Clozapine dihydrochloride			D₂ Receptor, Ki: 75 nM
Haloperidol-d₄-1			D₂ Receptor				98.0%
Pramipexole-d₅ dihydrochloride			D₂ Receptor	D₃ Receptor	D₄ Receptor
Flupentixol		D₁ Receptor	D₂ Receptor
1192U90			D₂ Receptor
Clozapine hydrochloride			D₂ Receptor, Ki: 75 nM
SB-414796			D₂ Receptor, Ki: 400 nM	D₃ Receptor, Ki: 4 nM
Tiapride			D₂ Receptor, IC₅₀: 110-320 nM	D₃ Receptor, IC₅₀: 180 nM
(Z)-Flupenthixol decanoate		D₁ Receptor	D₂ Receptor
PNU-96415E					D₄ Receptor
Raclopride tartrate		D₁ Receptor, Ki: 18000 nM	D₂ Receptor, Ki: 1.8 nM	D₃ Receptor, Ki: 3.5 nM	D₄ Receptor, Ki: 2400 nM
Dopamine D3 receptor ligand-6				D₃ Receptor
FR 64822			D₂ Receptor
Haloperidol-d₄ N-Oxide			D₂ Receptor
Risperidone mesylate			D₂ Receptor, Ki: 5.9 nM
U-101958 maleate			D₂ Receptor, IC₅₀: 1980 nM	D₃ Receptor, IC₅₀: 552 nM	D₄ Receptor, IC₅₀: 2.7 nM
ADX-10061		D₁ Receptor, Ki: 5.8 nM	D₂ Receptor, Ki: > ＞10 000 nM
BRD5814			D₂ Receptor
Metopimazine-d₆			D₂ Receptor
Iloperidone hydrochloride		Rat D₁ Receptor, Ki: 546 nM Human D₁ Receptor, Ki: 216 nM	Rat D₂ Receptor, Ki: 54 nM	Human D₃ Receptor, Ki: 7.1 nM	Human D₄ Receptor, Ki: 25 nM	Human D₅ Receptor, Ki: 319 nM
Dopamine D3 receptor ligand-5		D₁ Receptor, Ki: 4600 nM	D₂ Receptor, Ki: 2.85 nM	D₃ Receptor, Ki: 0.14 nM	D₄ Receptor, Ki: 756 nM
FAUC-312		Dopamine D1 receptor, Ki: 29000 nM	Dopamine D2 receptor, Ki: 25000 nM	Dopamine D3 receptor, Ki: 13000 nM	Dopamine D4 receptor, Ki: 1.5 nM
Sumanirole			D₂ Receptor
Pardoprunox			D₂ Receptor, pEC₅₀: 8	D₃ Receptor, pEC₅₀: 9.2
7-Hydroxy-PIPAT				D₃ Receptor, Ki: 0.99 nM
Thioridazine-d3 2-Sulfone				D₃ Receptor
Sarizotan dihydrochloride				Human D₃ Receptor, IC₅₀: 6.8 nM
Blonanserin-d₅			D₂ Receptor
ABT-724					D₄ Receptor	D₅ Receptor
Pimozide-d₅ N-Oxide		D₁ Receptor		D₃ Receptor
Abaperidone			D₂ Receptor, IC₅₀: 17 nM
NRA-0160				D₃ Receptor, Ki: 39 nM	D₄ Receptor, Ki: 0.48 nM
ABT-670					D₄ Receptor
Melperone-d₄ hydrochloride			Human D₂ Receptor, Kd: 180 nM				99.84%
Ropinirole-d₄ hydrochloride			D₂ Receptor	D₃ Receptor	D₄ Receptor
Desethoxy Quetiapine dihydrochloride			D₂ Receptor, IC₅₀: 1330 nM
Melperone (Standard)			Human D₂ Receptor, Kd: 180 nM
SKF 83509			D₂ Receptor, Ki: 70.2 nM
Dexpramipexole-d₃ dihydrochloride				D₃ Receptor
Raclopride-d₅ hydrochloride				D₃ Receptor			99.82%
BL-1020 mesylate			D_2S Receptor, Ki: 0.062 nM D_2L Receptor, Ki: 0.066 nM
Clocapramine dihydrochloride hydrate			D₂ Receptor
(-)-GSK598809				D₃ Receptor
BP 897 hydrochloride			D₂ Receptor	D₃ Receptor			99.84%

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