2. GPCR/G Protein Neuronal Signaling
  3. Opioid Receptor
  4. Cyprodime hydrochloride

Cyprodime hydrochloride 是一种高度选择性的 μ 阿片受体 (μ-opioid receptor) 拮抗剂，对于 μ，δ 和 κ 阿片受体的 Ki 值分别为 5.4 nM，244.6 nM 和 2187 nM。Cyprodime hydrochloride 具有抗抑郁样作用。

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Cyprodime hydrochloride Chemical Structure

Cyprodime hydrochloride Chemical Structure

CAS No. : 2387505-50-0

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Other Forms of Cyprodime hydrochloride:

Cyprodime hydrochloride 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Cyprodime hydrochloride is a highly selective μ-opioid receptor antagonist with Ki values of 5.4 nM, 244.6 nM and 2187 nM for μ-, δ- and κ-opioid receptors, respectively. Cyprodime hydrochloride has anti-depressant-like effect[1][2].

IC50 & Target

Ki: 5.4 nM (μ-opioid), 244.6 nM (δ-opioid) and 2187 nM (κ-opioid)[1]
体外研究
(In Vitro)

Cyprodime hydrochloride has Ki values of 8.1 nM and 26.6 nM for μ-opioid receptor in rat brain (Wistar) and guinea pig brain[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Cyprodime hydrochloride 相关抗体:
体内研究
(In Vivo)

Cyprodime hydrochloride (3, 10 mg/kg; i.p.; 60 min prior to test) significantly increases immobility time in the forced swimming test (FST) with higher dose of 10 mg/kg. Cyprodime hydrochloride increases the grooming time[2].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Male NMRI mice aged 21-25 days and weighing 10-12 g[2]
Dosage: 3, 10 mg/kg
Administration: IP; 60 min prior to test
Result: Significantly increased immobility time in the forced swimming test (FST) with higher dose of 10 mg/kg.
分子量

391.93

Formula

C22H30ClNO3
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Cyprodime hydrochloride 相关分类

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Cyprodime2387505-50-0Opioid Receptoranti-depressantimmobilitytimeforcedswimmingdepressantInhibitorinhibitorinhibit

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