1. Epigenetics
  2. Histone Demethylase
  3. LSD1-IN-22

LSD1-IN-22 是一种有效的赖氨酸特异性去甲基化酶 1 (LSD1) 抑制剂,Ki 为 98 nM。LSD1-IN-22 对某些癌细胞具有抗增殖活性。

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LSD1-IN-22 Chemical Structure

LSD1-IN-22 Chemical Structure

CAS No. : 2821068-05-5

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  • 生物活性

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生物活性

LSD1-IN-22 is a potent Lysine-specific demethylase 1 (LSD1) inhibitor with a Ki value of 98 nM. LSD1-IN-22 has anti-proliferative activity against certain cancer cells[1].

IC50 & Target

KDM1/LSD1

 

体外研究
(In Vitro)

LSD1-IN-22 (compound 7t) has anti-proliferative activity against CCRF-CEM, Jurkat and hERG cells[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Cell Proliferation Assay[1]

Cell Line: CCRF-CEM, Jurkat and hERG
Concentration: 0-50 μM
Incubation Time: 72 h
Result: Exhibited anti-proliferative activity against CCRF-CEM, Jurkat and hERG cells with IC50s of 23±0.8 μM, 26±1.7 μM and 7.7±1.3 μM.
分子量

248.07

Formula

C9H8BrF2N

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
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  • 稀释计算器

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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产品名称:
LSD1-IN-22
目录号:
HY-151191
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