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1061556-49-7

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抑制剂 & 激动剂

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Cat. No. Product Name Target Research Area Chemical Structure
  • HY-P1424A

    Potassium Channel
    Lei-Dab7 TFA is a high affinity, selective KCa2.2 (SK2) channel blocker (Kd=3.8 nM). Lei-Dab7 TFA exhibits >200-fold selectivity for KCa2.2 over KCa2.1, KCa2.3, KCa3.1, Kv and Kir2.1. Lei-Dab7 TFA increases theta-burst responses and increases LTP in rat hippocampal slices in vitro.
    Lei-Dab7 TFA
  • HY-P1424

    Potassium Channel Neurological Disease
    Lei-Dab7 是一种有效的选择性 SK2 (KCa2.2) 通道阻滞剂,Kd 为 3.8 nM。Lei-Dab7 在 KCa1、KCa3、Kv 和 Kir2.1 通道上显示低活性或无活性。
    Lei-Dab7

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