1. Epigenetics
  2. Histone Methyltransferase
  3. UNC2399

UNC2399 

目录号: HY-136188
产品使用指南

UNC2399,一种生物素化的 UNC1999,是选择性的 EZH2 降解剂,对 EZH2 具有很高的体外效力,IC50 值为 17 nM。

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UNC2399 Chemical Structure

UNC2399 Chemical Structure

CAS No. : 2412791-72-9

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Description

UNC2399, a biotinylated UNC1999, is a selective EZH2 degrader, maintaining high in vitro potency for EZH2, with an IC50 of 17 nM[1][2].

IC50 & Target[1]

EZH2

17 nM (IC50)

In Vitro

UNC2399 (1-1000 nM) displays high in vitro potency (IC50=17±2 nM) in the EZH2 radioactive biochemical assay[1].
UNC2399 (100 μM) enriches EZH2 from HEK293T cell lysates[1].

Molecular Weight

927.17

Formula

C₄₈H₆₆N₁₀O₇S

CAS No.

2412791-72-9

SMILES

CC(N1C2=CC(C(C=C3)=CN=C3N4CCN(CC4)C(CCOCCCOCCNC(CCCC[C@H]5[C@@H]6[C@@H](NC(N6)=O)CS5)=O)=O)=CC(C(NCC7=C(CCC)C=C(NC7=O)C)=O)=C2C=N1)C.[11]

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

UNC2399UNC 2399UNC-2399Histone MethyltransferasebiotinylatedUNC1999Inhibitorinhibitorinhibit

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产品名称:
UNC2399
目录号:
HY-136188
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