1. Signaling Pathways
  2. GPCR/G Protein
  3. Angiotensin Receptor
  4. Angiotensin Receptor Inhibitors

Angiotensin Receptor Inhibitors

AT1 Receptor

AT2 Receptor

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Angiotensin Receptor Inhibitors, Agonists, Antagonists, Modulators & Chemicals
Product Name AT1 Receptor AT2 Receptor Purity
Angiotensin II human
AT1 Receptor
AT2 Receptor
99.98%
Losartan
AT1 Receptor
  99.57%
Angiotensin II human acetate
AT1 Receptor
AT2 Receptor
99.81%
Telmisartan
AT1 Receptor
  99.79%
Nitrosoglutathione
AT1 Receptor
 
L-162537
AT1 Receptor, IC50: 1.7 nM
 
Valsartan
AT1 Receptor
  99.97%
Talfirastide
AT1 Receptor
  99.91%
Buloxibutid
AT1 Receptor, Ki: >10 μM
AT2 Receptor, Ki: 0.4 nM
98.94%
Losartan potassium
AT1 Receptor
  99.98%
Olmesartan
AT1 Receptor
  99.91%
A 779
AT1 Receptor
AT2 Receptor
99.12%
PD 123319 ditrifluoroacetate  
AT2 Receptor
99.82%
Olmesartan medoxomil
AT1 Receptor
  99.12%
TRV-120027
AT1 Receptor
  98.11%
Azilsartan
AT1 Receptor
  99.68%
Olodanrigan  
AT2 Receptor
98.89%
Talfirastide acetate
AT1 Receptor
  99.77%
TRV055
AT1 Receptor
  99.47%
Angiotensin III, human, mouse  
AT2 Receptor
98.26%
CGP-42112
AT1 Receptor
AT2 Receptor
99.84%
Fimasartan
AT1 Receptor
  99.60%
Azilsartan medoxomil
AT1 Receptor
  99.60%
TRV055 hydrochloride
AT1 Receptor
  98.88%
GSK1820795A
AT1 Receptor, IC50: 0.006 μM
  99.80%
Angiotensin II human TFA
AT1 Receptor
AT2 Receptor
98.84%
TRV-120027 TFA
AT1 Receptor
  99.69%
TRV056
AT1 Receptor
  99.91%
(Sar1,Ile4,8)-Angiotensin II
Angiotensin II Type 1
  99.75%
Tasosartan
AT1 Receptor
  99.32%
Losartan-d4
AT1 Receptor
  99.93%
ZD 7155(hydrochloride)
AT1 Receptor
  99.88%
(Sar1)-Angiotensin II
AT1 Receptor
  99.84%
Olmesartan-d4
AT1 Receptor
  98.83%
Olmesartan-d6
AT1 Receptor
  98.68%
PD 123177  
AT2 Receptor
98.14%
Valsartan-d9
AT1 Receptor
  99.33%
PD 123319  
AT2 Receptor
Olmesartan methyl ester
AT1 Receptor
 
Candesartan methyl ester  
AT2 Receptor, IC50: 66 nM
99.07%
Azilsartan medoxomil monopotassium
AT1 Receptor
  98.00%
Novokinin TFA  
AT2 Receptor
Olmesartan medoxomil-d6
AT1 Receptor
 
CI-996
AT1 Receptor
 
KRH-594
AT1 Receptor
 
EXP-7711
AT1 Receptor
 
CR 3834
AT1 Receptor
 
YM-358 hydrate potassium
Angiotensin II Type 1
 
GA-0056  
AT2 Receptor
EMD 66684
Angiotensin II Type 1, IC50: 0.7 nM
 
KR31173
AT1 Receptor, IC50: 3.27 nM
 
L-161638  
AT2 Receptor
LY 301875
Angiotensin II Type 1, pkB: 9.6
 
Ripisartan  
AT2 Receptor
AT2R antagonist 1  
AT2 Receptor
AT2R antagonist 2  
AT2 Receptor
L-163958
AT1 Receptor, IC50: 0.16 nM
AT2 Receptor, IC50: 0.12 nM
Olmesartan medoxomil (Standard)
AT1 Receptor
 
A-81282
AT1 Receptor, pA2: 9.64
 
rac-Olodanrigan
AT1 Receptor, IC50: 2918 nM
AT2 Receptor, IC50: 75.2 nM
CL-329167  
AT2 Receptor, IC50: 6 nM
UR-7247
AT1 Receptor
 
Elisartan
AT1 Receptor
 
TA-606  
AT2 Receptor