1. GPCR/G Protein
  2. Adenosine Receptor
  3. Derenofylline

Derenofylline (Synonyms: SLV 320)

目录号: HY-14858 纯度: >99.0%
产品使用指南

Derenofylline (SLV 320) 是一个有效的、选择性的、具有口服活性的腺苷A1 受体的拮抗剂,其对腺苷A1、A3 和A2A 受体的 Ki 值分别为 1 nM、200 nM 和 398 nM。Derenofylline可抑制心肌纤维化,降低蛋白尿,且不影响大鼠血压。

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Derenofylline Chemical Structure

Derenofylline Chemical Structure

CAS No. : 251945-92-3

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Description

Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. Derenofylline suppresses cardiac fibrosis and attenuates albuminuria without affecting blood pressure in rats[1].

IC50 & Target

Ki: 1 nM (adenosine A1 receptor)[1].

Clinical Trial
Molecular Weight

308.38

Formula

C₁₈H₂₀N₄O

CAS No.

251945-92-3

SMILES

O[C@H]1CC[C@H](NC2=C3C(NC=C3)=NC(C4=CC=CC=C4)=N2)CC1

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
References

Purity: >99.0%

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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产品名称:
Derenofylline
目录号:
HY-14858
需求量:

Derenofylline

Cat. No.: HY-14858