1. Screening Libraries
  2. GPCR/G Protein Compound Library

GPCR/G 蛋白化合物库 - GPCR/G Protein Compound Library

Cat. No.: HY-L006
Library Contents: XLSX PDF SDF

G 蛋白偶连受体 (GPCR) 是人类基因组中最大的一类膜蛋白,参与多种信号转导过程。信号分子与GPCR 结合,导致 G 蛋白的激活,并参与下一步的信号传递过程。GPCR 受体在机体内发挥着特别重要的作用,对这些受的进一步认识也会对现代医学产生一定的影响。事实上,研究人员预计,将有三分之一至一半数量的上市药物都是靶向 GPCR 受体的。GPCR 受体是药物开发中的一类主要靶点。

MCE 收录了 1105 种靶向 GPCRs 的小分子化合物,可以用于 GPCR 相关的不同研究及药物开发筛选。

GPCR/G Protein Compound Library
Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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  • Description

  • Product Details

  • Composition

  • Documentation

& Advantages

•   A unique collection of 1105 small molecules targeting G protein coupled receptors used in GPCR screening for various research and drug development projects.

•   Targets such as 5-HT Receptor, Dopamine Receptor, Opioid Receptor, Adrenergic Receptors, Cannabinoid Receptor, mGluR, ETA Receptor, etc.

•   The most successful class of drugable targets in the human genome and remain the most attractive family of targets.

•   All of the small molecules in the GPCR library are well characterized with biological and pharmaceutical activity. Some compounds have been approved by the FDA.

•   A powerful tool for discovering GPCR-based drugs that are the richest signal receptor targets for drug discovery.

•   Structurally diverse, medicinally active, and cell permeable.

•   Rich documentation with structure, IC50, and brief introduction.

•   NMR and HPLC validated to ensure the highest purity.

•   All compounds are in stock and continuously updated.

Product Details
A collection of 1105 GPCR/G Protein related compounds supplied as pre-dissolved DMSO solutions or Solid
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Blue ice

GPCR/G Protein Compound Library

Source: MedChem Express

Contents of GPCR/G Protein Compound Library


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GPCR/G Protein Compound Library

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