2. Metabolic Enzyme/Protease Immunology/Inflammation GPCR/G Protein Neuronal Signaling
  3. Lipoxygenase Histamine Receptor
  4. Linetastine

Linetastine  (Synonyms: 利奈他斯汀)

目录号: HY-123103
产品使用指南

摩尔计算器

Linetastine 是一种口服有效的 5-Lipoxygenase 抑制剂。Linetastine 具有抗组胺活性。Linetastine 抑制白三烯的产生并拮抗组胺的作用。Linetastine 抑制钙离子载体刺激的人白细胞释放白三烯 B4 和 C4。

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Linetastine Chemical Structure

Linetastine Chemical Structure

CAS No. : 159776-68-8

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Linetastine 相关抗体

Top Publications Citing Use of Products

查看 Lipoxygenase 亚型特异性产品:

查看所有亚型
5-LOX 12-LOX 15-LOX

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Linetastine is an orally active and potent 5-Lipoxygenase inhibitor. Linetastine shows antihistamine activity. Linetastine inhibits leukotriene production and antagonizes the effect of histamine. Linetastine inhibits the release of leukotrienes B4 and C4 from calcium ionophore-stimulated human leukocytes[1].

IC50 & Target

5-Lipoxygenase

 

Histamine Receptor

 

体内研究
(In Vivo)

在豚鼠中，Linetastine (1-10 mg/kg, 口服)可剂量依赖性地抑制组胺诱导的支气管收缩，且作用持续超过 24 小时[1]。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

584.70

Formula

C35H40N2O6
CAS 号
中文名称

利奈他斯汀
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Linetastine 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Linetastine159776-68-8利奈他斯汀LipoxygenaseHistamine ReceptorLOXInhibitorinhibitorinhibit

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