1. Protein Tyrosine Kinase/RTK
    JAK/STAT Signaling
  2. EGFR
  3. Khellin

Khellin 

目录号: HY-B1394
产品使用指南

Khellin 是一种自然产生的呋喃并色酮,是一种 EGFR 抑制剂,其 IC50 为 0.15 µM。Khelline 在体外具有抗增殖活性。Khellin 具有抗痉挛、舒张冠脉作用。

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Khellin Chemical Structure

Khellin Chemical Structure

CAS No. : 82-02-0

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Description

Khellin, a naturally occurring furochromone, is an EGFR inhibitor with an IC50 of 0.15 µM. Khelline has anti-proliferative activity in vitro. Khellin has antispasmodic and coronary vasodilator effects[1][2].

IC50 & Target

IC50: 0.15 µM (EGFR)[1]

In Vitro

Khelline exhibits anti-proliferative activity for MCF-7 cells and Hela cells[1].
Khellin causes total relaxation of both NA- and K+-contractions and a change in external calcium concentration[2].

Molecular Weight

260.24

Formula

C₁₄H₁₂O₅

CAS No.

82-02-0

中文名称

呋喃并色酮

SMILES

O=C1C=C(C)OC2=C(OC)C(OC=C3)=C3C(OC)=C12

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

KhellinEGFREpidermal growth factor receptorErbB-1HER1vascularsmoothmusclevitiligoanalgesicInhibitorinhibitorinhibit

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产品名称:
Khellin
目录号:
HY-B1394
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