1. Signaling Pathways
  2. PROTAC
  3. PROTACs
  4. PROTACs Inhibitors

PROTACs Inhibitors

von Hippel-Lindau (VHL)

Cereblon

MDM2

cIAP1

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PROTACs Degraders, Controls & Inhibitors
Product Name von Hippel-Lindau (VHL) Cereblon MDM2 cIAP1 Purity
FKBP12 PROTAC dTAG-13  
Cereblon
    99.89%
dBET6  
Cereblon
    99.92%
dAurAB5  
Cereblon
    99.03%
TO-1187 TFA  
Cereblon
    98.41%
DT2216
VHL
      99.97%
dBET1  
Cereblon
    99.24%
ACBI1
VHL
      99.92%
SD-36  
Cereblon
    99.73%
AK-1690  
Cereblon
    99.91%
dCBP-1  
Cereblon
    99.37%
MD-224    
MDM2, IC50: 1 nM
  99.60%
BSJ-4-116  
Cereblon
    99.87%
Bexobrutideg  
Cereblon
    99.33%
Setidegrasib
VHL
      99.65%
MS67
VHL
      98.73%
ZXH-3-26  
Cereblon
    98.90%
ARCC-4
VHL
      99.88%
LC-2
VHL
      98.48%
ACBI2
VHL, EC50: 7 nM
      99.76%
CFT8634  
Cereblon
    98.10%
GNE-987
VHL
      99.98%
PROTAC-O4I2  
Cereblon
    99.56%
MS4078  
Cereblon
    99.72%
PROTAC CBP/P300 Degrader-1  
Cereblon
    99.91%
PROTAC CDK2/9 Degrader-1  
Cereblon
    99.85%
XY028-140  
Cereblon
    98.52%
Tagarafdeg  
Cereblon
    99.41%
BSJ-03-123  
Cereblon
    99.19%
FKBP12 PROTAC dTAG-7  
Cereblon
    99.47%
TL12-186  
Cereblon
    99.63%
Nampt degrader-2
VHL
      99.41%
INY-03-041  
Cereblon
    99.74%
Seldegamadlin  
Cereblon
    98.53%
PROTAC α-Synuclein/Tau degrader 1  
Cereblon (α-Synuclein Ligand)
    99.28%
PROTAC KRAS G12D degrader 1
VHL
      98.32%
PIK5-12d
VHL
      99.90%
JET-209  
Cereblon
    98.07%
MS4322
VHL
Cereblon
MDM2
  99.14%
SJF-0628
VHL
      99.90%
JB170  
Cereblon
    98.97%
SJ10542  
Cereblon
    99.32%
MT-802  
Cereblon
    98.35%
LLC0424  
Cereblon
    98.42%
YD23  
Cereblon
    98.80%
PROTAC RIPK degrader-2
VHL
      99.89%
PROTAC K-Ras Degrader-1  
Cereblon
    99.90%
CP-10  
Cereblon
    98.41%
PROTAC HSP90 degrader BP3  
Cereblon
    99.54%
BMS-986458  
Cereblon
    99.65%
PROTAC SGK3 degrader-1
VHL
      99.89%
CRBN-6-5-5-VHL  
Cereblon, DC50: 1.5 nM
    99.45%
JH-XI-10-02  
Cereblon
    99.73%
FKBP12 PROTAC RC32  
Cereblon
    98.58%
BI-3663  
Cereblon
    99.84%
GMB-475
VHL
      98.69%
PROTAC NCOA4 degrader-1
VHL
      99.42%
MS8847
VHL
      99.78%
MS154  
Cereblon
    99.71%
ARD-266
VHL
      99.94%
TL13-112  
Cereblon, IC50: 2.4 μM
    98.01%
PROTAC CRBN Degrader-1
VHL
Cereblon
    98.77%
GBD-9  
Cereblon
Cereblon
    99.76%
TMX-4153
VHL
      98.96%
Homo-PROTAC cereblon degrader 1  
Cereblon
    99.66%
dFKBP-1  
Cereblon
    98.00%
PROTAC EED degrader-2
VHL
      99.90%
MS170  
CRBN-DDB1
    98.68%
MG-277  
Cereblon
    98.68%
ARD-69
VHL
      99.61%
ZXH-4-130 TFA
VHL
      99.71%
PROTAC MDM2 Degrader-3    
MDM2
 
PROTAC PD-1/PD-L1 degrader-1  
Cereblon
    99.52%
PROTAC KRAS G12C degrader-1  
Cereblon
    99.15%
PROTAC Bcl-xL degrader-2
VHL
      98.23%
SIAIS178
VHL
      99.36%
PROTAC MDM2 Degrader-2    
MDM2
 
SJF620  
Cereblon
    98.98%
Tz-Thalidomide  
Cereblon
    98.60%
PROTAC BRD9 Degrader-1  
CRBN-DDB1, IC50: 48.9 nM
    99.16%
XZ739  
Cereblon
    99.06%
PROTAC IRAK4 degrader-1  
Cereblon
    99.77%
PROTAC FKBP Degrader-3
VHL
      99.48%
PROTAC EGFR degrader 9  
Cereblon
    98.35%
MD-222    
MDM2
  99.81%
PROTAC EZH2 Degrader-2    
MDM2
  99.78%
SHP2-D26 isomer-1
VHL
      99.76%
SJF-1521
VHL
      99.65%
PROTAC PARP1 degrader    
MDM2
  99.74%
SR-1114  
Cereblon
    99.04%
PROTAC EED degrader-1
VHL
      98.27%
PZ703b
VHL
      98.00%
PROTAC ERRα Degrader-3
VHL
      98.82%
PROTAC ERα Degrader-2      
cIAP1
98.92%
PROTAC RAR Degrader-1      
cIAP1
TD-165  
Cereblon, DC50: 20.4 nM
    98.08%
SJFα
VHL
      99.61%
PROTAC ER Degrader-4
VHL
      98.78%
MS4077  
Cereblon
    99.66%
FMF-06-098-1
VHL
      98.77%
MZP-54
VHL
      98.03%
Homo-PROTAC pVHL30 degrader 1
VHL
      99.40%
TL13-12  
Cereblon, IC50: 1.2 μM
    98.16%
PROTAC RIPK degrader-6  
Cereblon
    99.01%
INY-03-041 trihydrochloride  
Cereblon
    98.44%
CCT367766 formic  
CRBN-DDB1, IC50: 490 nM
    98.10%
ARD-2051  
Cereblon
    98.57%
DD-03-171  
Cereblon
    98.72%
HDAC6 degrader-3  
Cereblon
    98.60%
SK2188  
Cereblon
   
SIA​​IS039  
Cereblon
    99.68%
PROTAC MDM2 Degrader-1    
MDM2
  98.11%
PROTAC PD-L1 degrader-1  
Cereblon, Kd: 131.77 μM
    98.03%
PROTAC BRD9 Degrader-7  
Cereblon
    99.29%
ARD-61
VHL
      99.57%
MS4322 (isomer)
VHL
Cereblon
MDM2
  99.22%
SD-436  
Cereblon
    98.27%
OARV-771
VHL
      98.77%
PROTAC ERRα Degrader-1    
MDM2
  98.22%
TD-428  
Cereblon
    98.81%
UBX-382  
Cereblon
   
PROTAC EGFR degrader 11  
CRBN-DDB1, Ki: 36 nM
    99.20%
Thalidomide-NH-CBP/p300 ligand 2  
Cereblon
    98.55%
MI-389  
Cereblon
    99.34%
PROTAC SMARCA2/4 degrader-38
VHL
      99.46%
WH-10417-099  
Cereblon
    98.14%
PROTAC EGFR degrader 15  
Cereblon
   
XY-06-007  
Cereblon
    98.9%
PROTAC AR Degrader-4      
cIAP1
PROTAC AR Degrader-4 TFA      
cIAP1
99.26%
DP-C-4  
Cereblon
    98.15%
SJF620 hydrochloride  
Cereblon
    99.28%
MS33
VHL
     
PROTAC K-Ras Degrader-5  
Cereblon
   
dCDK9-202  
Cereblon
   
DGY-09-192
VHL
      99.50%
TO-1187  
Cereblon
   
JCS-1
VHL
      99.38%
PROTAC EGFR degrader 14
VHL
     
SJFδ
VHL
     
PROTAC HER2 degrader-1  
CRBN-DDB1
    98.0%
JP-163-16  
Cereblon
   
PROTAC HDAC degrader-2  
Cereblon
   
FPP29
VHL
     
AF151
VHL
     
MI1013  
Cereblon
   
PROTAC ERRα Degrader-2    
MDM2
 
MS98
VHL
     
PROTAC BRD4 Degrader-2  
Cereblon
   
MD-4251    
MDM2
 
CCT367766  
CRBN-DDB1, IC50: 490 nM
   
PROTAC SMARCA2 degrader-30  
Cereblon
   
JB300  
Cereblon
   
PROTAC Bcl-xL degrader-3
VHL
     
PROTAC SARS-CoV-2 RdRp Degrader-1  
Cereblon
   
PROTAC BTK Degrader-12  
Cereblon
   
PROTAC DAPK1 Degrader-1  
Cereblon
   
PZ671  
Cereblon
   
JPS004
VHL
     
PROTAC BRD4 Degrader-40  
Cereblon
   
PROTAC SMARCA2 degrader-27
VHL
     
(S)-GNE-987
VHL
     
Abd110  
Cereblon
   
PROTAC ERα Degrader-12
VHL
     
Naph-Se-TMZ  
Cereblon
   
TAT-PiET-PROTAC
VHL
     
PROTAC CDK4/6/9 degrader 1  
Cereblon
   
PROTAC FLT-3 degrader 4  
Cereblon
   
PROTAC BRD4 Degrader-34
VHL
     
PROTAC ERα Degrader-13
VHL
     
YTHu78  
Cereblon
   
PROTAC EGFR degrader 16  
Cereblon
   
SJ46420
VHL
     
CST651
VHL
     
MS910  
Cereblon
   
JQ1-S(GlcNAc)Cq  
Cereblon
   
SA-PA  
Cereblon
   
ZXH-4-130
VHL
     
CH091138
VHL
     
PROTAC FLT3/CHK1 Degrader-1  
Cereblon
   
PROTAC SGK3 degrader-2
VHL
     
Psa-AR  
Cereblon
   
PROTAC FAK degrader 3  
Cereblon
   
MS44
VHL
     
PROTAC HDAC6 degrader 8  
Cereblon
   
PROTAC sEH-degrader-3  
Cereblon
   
PROTAC K-Ras Degrader-6  
Cereblon
   
dASK1  
Cereblon
   
PROTAC Bcl-xL degrader-1      
cIAP1
PROTAC PI3Kα degrader-1  
Cereblon
   
NU223612  
Cereblon
   
UNC9036
VHL
     
PROTAC tubulin-Degrader-1  
Cereblon
   
SIAIS562055  
Cereblon
   
PROTAC sEH degrader-2  
Cereblon
   
TQ-3959  
Cereblon
   
BT-O2C  
Cereblon
   
SD-2301
VHL
     
PROTAC BRAF-V600E degrader-2  
Cereblon
   
C199
VHL
     
PROTAC FLT3/JAK2/BRD4 Degrader-1  
Cereblon
   
PROTAC MDM2 Degrader-4    
MDM2
 
PROTAC RIPK1 Degrader-1
VHL
     
PROTAC HPK1 Degrader-5  
Cereblon
   
PROTAC TG2 degrader-1
VHL
     
DDD2
VHL
     
PROTAC RET Degrader 1  
Cereblon
   
LYA914  
Cereblon
   
PROTAC FLT-3 degrader 5  
Cereblon
   
PROTAC BCL6/IKZF1/3 Degrader-1  
Cereblon
   
RIP2 Kinase Inhibitor 4      
cIAP1
SA-VA
VHL
     
PROTAC G9a/GLP degrader 1
VHL
     
PROTAC FTO degrader 1
VHL
     
PROTAC BTK/IKZF1/3 Degrader-1  
Cereblon
   
LAG-3 PROTAC-1  
Cereblon
   
DeFer-2
VHL
     
PROTAC EGFR degrader 10  
CRBN-DDB1, Ki: 37 nM
   
PROTAC SOS1 degrader-3  
Cereblon
   
L134  
Cereblon
   
PROTAC SMARCA2 degrader-3  
Cereblon
   
PROTAC BRD4 Degrader-39
VHL
     
FIP22  
Cereblon
   
PROTAC JAK2 degrader-1  
Cereblon
   
PROTAC AR Degrader-10  
CRBN-DDB1
   
PROTAC BRD2/BRD4 degrader-1  
Cereblon
   
PROTAC ER Degrader-11  
Cereblon
   
PROTAC HBeAg degrader-1
VHL